Compile Data Set for Download or QSAR
maximum 50k data
Found 34 of ic50 data for polymerid = 50000014
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50052524((S)-N-((S)-1-{[(S)-1-({[(S)-1-((S)-1-Carbamoyl-3-m...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50050641(CHEMBL45340 | PD-161182 | [(R)-2-(2,3-Difluoro-phe...)
Affinity DataIC50:  30nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030146(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Tle-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  65nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50194575(CHEMBL219162 | N'-(3-methoxy-2-phenyl-quinoline-4-...)
Affinity DataIC50:  66nMAssay Description:Binding affinity to rat NK3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50050652(CHEMBL47146 | PD-160946 | [(R)-2-(2-Fluoro-phenyl)...)
Affinity DataIC50:  83nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030158(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Flg-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  91nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030163(Arg-Pro-Lys-Pro-Gln-Gln-Phe-(2S,3S)Ing-Flg-Leu-Met...)
Affinity DataIC50:  110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50407164(CHEMBL2115376)
Affinity DataIC50:  110nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030154(Arg-Pro-Lys-Pro-Gln-Gln-(2S,3S)Bfi-Phe-Gly-Leu-Met...)
Affinity DataIC50:  120nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  130nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030166(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Pen(S-Me)-Gly-Leu-Met ...)
Affinity DataIC50:  170nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50407161(CHEMBL2114443)
Affinity DataIC50:  180nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030153(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Pen(SO2-Me)-Gly-Leu-Me...)
Affinity DataIC50:  190nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030165(Arg-Pro-Lys-Pro-Gln-Gln-Tic-Phe-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  520nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030170(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Met-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  1.20E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030164(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Flg-Pro-Leu-Met | CHEM...)
Affinity DataIC50:  1.30E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50050649(CHEMBL444832 | {(S)-1-[(R)-1-Methyl-2-phenyl-1-(7-...)
Affinity DataIC50:  1.73E+3nMAssay Description:Inhibitory activity against cloned human Tachykinin receptor 3 in CHO cells labeled with [125I][MePhe7]-NKBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030157(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Hph-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  1.90E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50407163(CHEMBL2114442)
Affinity DataIC50:  2.10E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50407162(CHEMBL2115375)
Affinity DataIC50:  2.20E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030160(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Dip-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  2.20E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50050642(CHEMBL296014 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  2.79E+3nMAssay Description:In vitro inhibitory activity against senktide-evoked increases in intracellular calcium levels in cloned human Tachykinin receptor 3 in CHO cell line...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030152(Arg-Pro-Lys-Pro-Gln-Gln-Flg-Phe-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  3.10E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50002462(1,3-Diethyl-2-[3-(1,3,3-trimethyl-1,3-dihydro-indo...)
Affinity DataIC50:  3.30E+3nMAssay Description:Binding affinity of compound was evaluated towards tachykinin receptor 3 by using radioligand [1261]eledoisin in rat cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030167(Arg-Pro-Lys-Pro-Gln-Gln-Met-Phe-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  7.40E+3nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030161(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Pro-Leu-Met | CHEM...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030159(Arg-Pro-Lys-Pro-Gln-Gln-Hph-Phe-Gly-Leu-Met | CHEM...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030155(Arg-Pro-Lys-Pro-Gln-Gln-deltaZPhe-Phe-Gly-Leu-Met ...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030148(Arg-Pro-Lys-Pro-Gln-Gln-[D-2Ing]-Phe-Gly-Leu-Met |...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030150(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Dip-Pro-Leu-Met | CHEM...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030147(Arg-Pro-Lys-Pro-Gln-Gln-2Ing-Phe-Gly-Leu-Met | CHE...)
Affinity DataIC50: >1.00E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030155(Arg-Pro-Lys-Pro-Gln-Gln-deltaZPhe-Phe-Gly-Leu-Met ...)
Affinity DataIC50:  1.17E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030156(Arg-Pro-Lys-Pro-Gln-Gln-Dip-Phe-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  1.70E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuromedin-K receptor(Rattus norvegicus)
Cambridge University Forvie Site

Curated by ChEMBL
LigandPNGBDBM50030168(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Tic-Gly-Leu-Met | CHEM...)
Affinity DataIC50:  1.80E+4nMAssay Description:Concentration required to inhibit the specific binding of [125I]BH-ELE to Neurokinin-3 (NK-3) receptor in rat brain synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed